41863-58-5Relevant articles and documents
Easy access to drug building-blocks through benzylic C-H functionalization of phenolic ethers by photoredox catalysis
Brandhofer, Tobias,Derdau, Volker,García Manche?o, Olga,Méndez, María,P?verlein, Christoph,Stinglhamer, Martin
supporting information, p. 6756 - 6759 (2021/07/13)
A visible light-mediated photocatalyzed C-C-bond forming method for the benzylic C-H functionalization of phenolether containing synthetic building blocks based on a radical-cation/deprotonation strategy is reported. This method allows the mild, selective generation of benzyl radicals in phenolic complex molecules and drug-like compounds, providing new entries in synthetic and medicinal chemistry.
Epimerization-free block synthesis of peptides from thioacids and amines with the sanger and mukaiyama reagents
Crich, David,Sharma, Indrajeet
supporting information; experimental part, p. 2355 - 2358 (2009/08/19)
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On the fate of the tryptophan stereocenter during the synthesis of hexacyclic analogues of N-acetylardeemin
Caballero, Esmeralda,Avendano, Carmen,Menendez, J. Carlos
, p. 3025 - 3038 (2007/10/03)
The reaction between 6-acetyl-3-alkyl-1-ethoxy-3,4,5a,6,11,11a- hexahydro-10bH-pyrazino-[2',1'-5,1]pyrrolo-[2,3-b]indole-1,4-diones and anthranilic acid was studied from a stereochemical point of view. Various degrees of epimerization of the tryptophan an
