4921-87-3Relevant articles and documents
GUANIDINE COMPOUNDS, AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5 RECEPTORS
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Page/Page column 74, (2010/02/13)
The invention relates to guanidine compounds of general formula (I), corresponding enantiomeric, diastereomeric, and/or tautomeric forms thereof, and pharmaceutically acceptable salts thereof. The invention further relates to the use of guanidine compounds as binding partners for 5-HT5 receptors in order to treat diseases modulated by 5-HT5 receptor activity, especially treat neurodegenerative and neuropsychiatric disorders and the signs, symptoms, and malfunctions associated therewith.
Synthesis and Antiinflammatory Activity of Some 5-Thiazoleacetic Acids
Sawhney, S. N.,Dhindsa, G. S.,Singh, S. P.
, p. 1044 - 1049 (2007/10/02)
Four series of 5-thiazoleacetic acids (I, II, III and IV) have been synthesized for evaluation as potential antiinflammatory agents.Compounds of the series I, II and IV have been prepared by the condensation of various β-aroyl-β-bromopropionic acids (VIII