5220-02-0 Usage
Description
DIAZEPAM RELATED COMPOUND B (25 MG) (3-AMINO-6-CHLORO-1-METHYL-4-PHENYLCARBOSTYRIL) is a chemical compound that is identified as an impurity in the synthesis of Diazepam, a well-known anxiolytic, muscle relaxant, and anticonvulsant medication. DIAZEPAM RELATED COMPOUND B (25 MG) (3-AMINO-6-CHLORO-1-METHYL-4-PHENYLCARBOSTYRIL) is characterized by its molecular structure, which includes an amino group, a chloro substituent, and a methyl group attached to a phenylcarbostyril backbone.
Uses
Used in Pharmaceutical Industry:
DIAZEPAM RELATED COMPOUND B (25 MG) (3-AMINO-6-CHLORO-1-METHYL-4-PHENYLCARBOSTYRIL) is used as an impurity in the synthesis of Diazepam (D416855) for the following reasons:
1. As an anxiolytic: It contributes to the development of medications that help alleviate anxiety and stress-related disorders.
2. As a muscle relaxant (skeletal): It plays a role in the creation of drugs that can help relax skeletal muscles, providing relief from muscle spasms and pain.
3. As an anticonvulsant: It is involved in the synthesis of medications that help prevent and control seizures, offering support to individuals with epilepsy and other seizure disorders.
Synthesis Reference(s)
The Journal of Organic Chemistry, 38, p. 449, 1973 DOI: 10.1021/jo00943a008
Check Digit Verification of cas no
The CAS Registry Mumber 5220-02-0 includes 7 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 4 digits, 5,2,2 and 0 respectively; the second part has 2 digits, 0 and 2 respectively.
Calculate Digit Verification of CAS Registry Number 5220-02:
(6*5)+(5*2)+(4*2)+(3*0)+(2*0)+(1*2)=50
50 % 10 = 0
So 5220-02-0 is a valid CAS Registry Number.
InChI:InChI=1/C16H13ClN2O/c1-19-13-8-7-11(17)9-12(13)14(15(18)16(19)20)10-5-3-2-4-6-10/h2-9H,18H2,1H3
5220-02-0Relevant articles and documents
Chemical transformations of 3-amino-2-quinolones
Asis, Silvia E.,Bruno, Ana M.,Dominici, Diego A.,Bollini, Mariela,Gaozza, Carlos H.
, p. 107 - 112 (2007/10/03)
In order to find new antimalarial drugs, an exploration about the chemical properties of the starting compounds 3-amino-6-chloro-4-phenyl-1H-quinolin-2-one (1) and 3-amino-4-methyl-1H-quinolin-2-one (2) was developed. Acylation with acyl chloride, sulfony
Synthesis of Pyridinium Heterocyclic Ylides. Degradation of the Pyridinium Group
Esteve, Marta E.,Gaozza, Carlos H.
, p. 1061 - 1063 (2007/10/02)
The synthesis of pyridinium-quinolone chlorides and ylides, a pyridinium-methylquinazolone ylide, 9-pyridinium acridine chloride, and their behaviour by treatment by boiling aniline are described.
The Conversion of 2-(2-Chloroacetamido)benzophenones into 2,3-Dihydro-2-oxo-1,4-benzodiazepines. Part I. With Ammonia
Clarke, George M.,Lee, J. Barry,Swinbourne, Frederick J.,Williamson, Basil
, p. 4745 - 4761 (2007/10/02)
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