61570-89-6Relevant articles and documents
Stereoselective and Site-Specific Allylic Alkylation of Amino Acids and Small Peptides via a Pd/Cu Dual Catalysis
Huo, Xiaohong,He, Rui,Fu, Jingke,Zhang, Jiacheng,Yang, Guoqiang,Zhang, Wanbin
supporting information, p. 9819 - 9822 (2017/08/02)
We report a stereoselective and site-specific allylic alkylation of Schiff base activated amino acids and small peptides via a Pd/Cu dual catalysis. A range of noncoded α,α-dialkyl α-amino acids were easily synthesized in high yields and with excellent enantioselectivities (up to >99% ee). Furthermore, a direct and highly stereoselective synthesis of small peptides with enantiopure α-alkyl or α,α-dialkyl α-amino acids residues incorporated at specific sites was accomplished using this dual catalyst system.
One-pot liquid-phase synthesis of DSIP and 5-phe-DSIP using fluoren-9-yl-methoxycarbonyl-protected amino acid pentafluorophenyl esters
Wang,Xu
, p. 845 - 846 (2007/10/02)
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Rapid peptide synthesis in liquid phase. Preparation of angiotensin II and delta-sleep-inducing peptide by the 'hold-in' solution method
Nozaki,Muramatsu
, p. 2165 - 2168 (2007/10/02)
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