625850-78-4Relevant articles and documents
Synthesis and structure-activity relationship of novel benzoxazole derivatives as melatonin receptor agonists
Sun, Li-Qiang,Chen, Jie,Bruce, Marc,Deskus, Jeffrey A.,Epperson, James R.,Takaki, Katherine,Johnson, Graham,Iben, Lawrence,Mahle, Cathy D.,Ryan, Elaine,Xu, Cen
, p. 3799 - 3802 (2007/10/03)
A series of benzoxazole derivatives was synthesized and evaluated as melatoninergic ligands. The binding affinity of these compounds for human MT1 and MT2 receptors was determined using 2-[ 125I]-iodomelatonin as the radio