628323-61-5Relevant articles and documents
Imidazo[1,2-a]pyrimidines as functionally selective GABAA ligands
Blackaby, Wesley P.,Atack, John R.,Bromidge, Frances,Castro, Jose L.,Goodacre, Simon C.,Hallett, David J.,Lewis, Richard T.,Marshall, George R.,Pike, Andrew,Smith, Alison J.,Street, Leslie J.,Tattersall, David F. D.,Wafford, Keith A.
, p. 1175 - 1179 (2006)
Imidazo[1,2-a]pyrimidines are GABAA receptor benzodiazepine binding site ligands which can exhibit functional selectivity for the α3 subtype over the α1 subtype. SAR studies to optimize this functional selectivity are desc
