690646-06-1Relevant articles and documents
Systematic variation of the benzoylhydrazine moiety of the GluN2A selective NMDA receptor antagonist TCN-201
Schreiber, Julian A.,Müller, Sebastian L.,Westph?linger, Stefanie E.,Schepmann, Dirk,Strutz-Seebohm, Nathalie,Seebohm, Guiscard,Wünsch, Bernhard
supporting information, p. 259 - 269 (2018/09/18)
GluN2A containing N-methyl-D-aspartate receptors (NMDARs) are important ion channels in the central nervous system and highly involved in several different neurophysiological but also neuropathophysiological processes. However, current understanding of th
4-(Phenylsulfonamidomethyl)benzamides as potent and selective inhibitors of the 11β-hydroxysteroid dehydrogenase type 1 with efficacy in diabetic ob/ob mice
Zhang, Xu,Zhou, Zhou,Yang, Huaiyu,Chen, Junhua,Feng, Ying,Du, Lili,Leng, Ying,Shen, Jianhua
supporting information; experimental part, p. 4455 - 4458 (2010/04/05)
Selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) have considerable potential as treatments for type 2 diabetes. Presented herein are the syntheses, structure-activity relationships, and efficacy evaluation of 4-(phenylsulfonamido