74371-91-8Relevant articles and documents
Heteroannulation of arynes with N-aryl-α-aminoketones for the synthesis of unsymmetrical N-aryl-2,3-disubstituted indoles: An aryne twist of Bischler-Moehlau indole synthesis
Bunescu, Ala,Piemontesi, Cyril,Wang, Qian,Zhu, Jieping
, p. 10284 - 10286 (2013/10/22)
Reaction of 2-(trimethylsilyl)aryl triflates 1 with N-aryl-α-amino ketones 2 afforded N-aryl-2,3-disubstituted indoles in good to excellent yields with complete control of the substitution patterns. This methodology allowed for the first time a one-step s
Zirconium-catalyzed multistep reaction of hydrazines with alkynes: A non-fischer-type pathway to indoles
Gehrmann, Thorsten,Lloret Fillol, Julio,Scholl, Solveig A.,Wadepohl, Hubert,Gade, Lutz H.
supporting information; experimental part, p. 5757 - 5761 (2011/08/05)
Dominos at zirconium: A cascade of N-N and C-H scissions and C-C and C-N coupling steps in the coordination sphere of zirconium directly converts alkynes and hydrazines into indoles. The reaction pathway differs fundamentally from that of the Fischer indo
Thermal cyclization of N-trifluoroacetyl enehydrazines under mild conditions: A novel entry into the Fischer indole synthesis
Miyata, Okiko,Kimura, Yasuo,Muroya, Kanami,Hiramatsu, Hajime,Naito, Takeaki
, p. 3601 - 3604 (2007/10/03)
An efficient thermal cyclization of N-trifluoroacetyl enehydrazines for the synthesis of indoles is described.
