80167-52-8Relevant articles and documents
Synthesis and antifungal activity of N-(alkyl/aryl)-2-(3-oxo-1,4- benzothiazin-2-yl)acetamide
Gupta,Wagh
, p. 697 - 702 (2007/10/03)
A series of N-(alkyl/aryl)-2-(3-oxo-1,4-benzothiazin-2-yl)acetamide have been synthesized by condensation of substituted amines with maleic anhydride (MA) followed by cyclization with o-aminothiophenol (o-ATP). All the compounds have been screened for their antifungal activity against Tricophyton rubrum, Epidermophyton floccosum and Malassazia furfur. In the primary screening, some of the compounds exhibited appreciable activity. The structures of the synthesized compounds 7a-z have been established on the basis of elemental analysis and spectral data.
Reactions of Cyclic Anhydrides: Part V - Acid-catalysed Esterification of Maleanilic and Fumaranilic Acids and Evidence of Activation by Carboxamido Function
Patel, M. V.,Balasubramaniyan, V.
, p. 804 - 805 (2007/10/02)
Maleanilic and fumaranilic acids undergo acid catalysed esterification with methanol under very mild conditions.Intramolecular activation involving carboxamido group appears likely in this reactions.