82003-76-7Relevant articles and documents
Potential Affinity Labels for the Opiate Receptor Based on Fentanyl and Related Compounds
Maryanoff, Bruce E.,Simon, Eric J.,Gioannini, Theresa,Gorissen, H.
, p. 913 - 919 (2007/10/02)
Derivatives of fentanyl, 3-methylfentanyl, sufentanil, and lofentanil, possesing chemo- or photoaffinity functionalities, were synthesized as potential affinity reagents for the opiate receptor.Opiate receptor binding constants (IC50) were determined in c