864724-72-1Relevant articles and documents
SnCl2/RSH: A versatile catalytic system for the synthesis of 4-Alkylsulfanyl-indazole derivatives
Kouakou, Assoman,Chicha, Hakima,Rakib, El Mostapha,Gamouh, Ahmed,Hannioui, Abdellah,Chigr, Mohammed,Viale, Maurizio
, p. 86 - 95 (2015/10/20)
The treatment of alkylated nitro derivatives of indazole with stannous chloride in alkanethiol gave after coupling of the obtained amines with 4-methoxybenzenesulfonyl chloride in pyridine the new N-(4-Alkylsulfanylindazol-7-yl)-4-methoxybenzene sulfonamides via the nucleophilic substitution of hydrogen in position 4 of indazole, together with the expected 4-methoxy-N-(indazol-7-yl)-benzenesulfonamides. All the newly synthesized compounds have been characterized by elemental analysis and spectroscopic data.
New and efficient synthesis of bi- and trisubstituted indazoles
Bouissane, Latifa,El Kazzouli, Sa?d,Léger, Jean-Michel,Jarry, Christian,Rakib, El Mostapha,Khouili, Mostafa,Guillaumet, Gérald
, p. 8218 - 8225 (2007/10/03)
In this paper, the synthesis of bi- and trisubstituted indazoles was described. 4-Alkoxy-7-aminoprotected-indazole or 7-aminoprotected-indazole derivatives were prepared selectively using SnCl2 in alcohol or SnCl2 in ethyl acetate, r