870524-83-7Relevant articles and documents
Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors
Xu, Jinyou,Wei, Lan,Mathvink, Robert,He, Jiafang,Park, You-Jung,He, Huaibing,Leiting, Barbara,Lyons, Kathryn A.,Marsilio, Frank,Patel, Reshma A.,Wu, Joseph K.,Thornberry, Nancy A.,Weber, Ann E.
, p. 2533 - 2536 (2005)
anti-Substituted β-methylphenylalanine derived amides have been shown to be potent DPP-IV inhibitors exhibiting excellent selectivity over both DPP8 and DPP9. These are among the most potent compounds reported to date lacking an electrophilic trap. The mo