872471-89-1Relevant articles and documents
2-(Benzimidazol-2-yl)quinoxalines: A novel class of selective antagonists at human A1 and A3 adenosine receptors designed by 3D database searching
Novellino, Ettore,Cosimelli, Barbara,Ehlardo, Marina,Greco, Giovanni,Iadanza, Manuela,Lavecchia, Antonio,Rimoli, Maria Grazia,Sala, Annalisa,Da Settimo, Antonio,Primofiore, Giampaolo,Da Settimo, Federico,Taliani, Sabrina,La Motta, Concettina,Klotz, Karl-Norbert,Tuscano, Daniela,Trincavelli, Maria Letizia,Martini, Claudia
, p. 8253 - 8260 (2005)
The Cambridge Structural Database (CSD) was searched through two 3D queries based on substructures shared by well-known antagonists at the A1 and A3 adenosine receptors (ARs). Among the resulting 557 hits found in the CSD, we selecte