90562-37-1Relevant articles and documents
Synthesis of 1-acyl-3,4-dihydroquinazoline-2(1H)-thiones by cyclization of N-[2-(isothiocyanatomethyl)phenyl] amides generated in situ from N-[2-(azidomethyl)phenyl] amides
Kobayashi, Kazuhiro,Matsumoto, Naoki
, p. 923 - 930 (2014/08/05)
An efficient method for the preparation of 1-acyl-3,4-dihydroquinazoline- 2(1H)-thiones 5 has been developed. The reaction of N-[2-(azidomethyl)phenyl] amides 3, easily prepared by a three-step sequence starting with (2-aminophenyl)methanols, with Ph
CYCLIZATION OF N-(2-AMINOBENZYL) BENZYLAMINO-1-PHENYL-1-ETHANOLS AND DEBENZYLATION OF THE RESULTING TETRAHYDROISOQUINOLINE DERIVATIVES
Zara-Kaczian, Erzsebet,Deak, Gyula,Szoelloesy, Aron,Brlik, Janos
, p. 743 - 755 (2007/10/02)
Debenzylation reactions of 2-(o-aminobenzyl)-4-phenyl-1,2,3,4-tetrahydroisoquinolines (3a, b) and their N-acetyl derivatives (4a, b), obtained by the cyclization of N-(2-aminobenzyl)benzylamino-1-phenyl-1-ethanols (1), were studied.