916518-48-4Relevant articles and documents
sp3 C-H bond arylation directed by amidine protecting group: α-arylation of pyrrolidines and piperidines
Pastine, Stefan J.,Gribkov, Denis V.,Sames, Dalibor
, p. 14220 - 14221 (2006)
A new ruthenium-catalyzed direct sp3 C-H to C-C bond transformation is disclosed. Specifically, a method for the α-arylation of cyclic amines, containing either permanent (pyridine, pyrimidine) or removable (amidine) directing groups, is descri