925673-30-9Relevant articles and documents
C6-(N,N-butyl-methyl-heptanamide) derivatives of estrone and estradiol as inhibitors of type 1 17β-hydroxysteroid dehydrogenase: Chemical synthesis and biological evaluation
Cadot, Christine,Laplante, Yannick,Kamal, Fatima,Luu-The, Van,Poirier, Donald
, p. 714 - 726 (2007/10/03)
A series of estrone and estradiol derivatives having an N-butyl,methyl heptanamide side chain at C6-position were synthesized, tested as inhibitors of type 1 17β-HSD and assessed for their possible estrogenic activity. A better type 1 17β-HSD inhibition w