943240-70-8Relevant articles and documents
Design, synthesis, and structure-affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties
Cappelli, Andrea,Giuliani, Germano,Anzini, Maurizio,Riitano, Daniela,Giorgi, Gianluca,Vomero, Salvatore
, p. 6850 - 6859 (2008/12/21)
The substituent in position 2 of the quinoline nucleus of NK1 receptor ligands 5 has been constrained into different five-membered heterocyclic moieties in order to obtain information on the binding site pocket interacting with this apparently