1261352-34-4Relevant articles and documents
A new approach to desketoraloxifene analogs from oxygen-bearing 3-iodobenzo[b]thiophenes prepared via iodocyclization
Cho, Chul-Hee,Jung, Dai-Il,Larock, Richard C.
supporting information; experimental part, p. 6485 - 6488 (2011/02/22)
A formal total synthesis of the benzothiophene selective estrogen receptor modulator (SERM) desketoraloxifene and analogs has been accomplished from alkynes bearing electron-rich aromatic rings by electrophilic cyclization using I2. This approa