205582-88-3Relevant articles and documents
METHOD FOR PREPARATION OF 6-TRIFLUOROMETHYLPYRIDINE-3-CARBOXYLIC ACID DERIVATIVES FROM TRIFLUOROACETYLACETIC ACID
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Page/Page column 11, (2015/02/02)
The invention discloses a method for the preparation of 6- trifluoromethylpyridine-3-carboxylic acid derivatives (I) from trifluoroacetylacetic acid (II) and orthoesters (III), and their use for the preparation of pharmaceutical, chemical or agro-chemical products.
Method for preparation of 6-trifluoromethylpyridine-3-carboxylic acid derivatives
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Paragraph 0043, (2014/12/09)
The invention discloses a method for the preparation of substituted 6-trifluoromethylpyridine-3-carboxylic acid derivatives starting from 1,1,1-trifluoroacetone or from synthetic equivalents of 1,1,1-trifluoroacetone.
Triazolopyridine cannabinoid receptor 1 antagonists
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Page/Page column 78, (2008/06/13)
The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents, and methods of treatment using the compounds according to Formula I both alone and in combination with one or more additional therapeutic agents. The compounds have the following general formula: including all prodrugs, solvates, pharmaceutically acceptable salts and stereoisomers, wherein R1, R2, R3, R4 and R5 are described herein.