103825-24-7Relevant articles and documents
Cholecystokinin antagonists. Synthesis and biological evaluation of 3-substituted benzolactams
Parsons,Patchett,Holloway,Smith,Davidson,Lotti,Chang
, p. 1681 - 1685 (1989)
A series of 1,3-substituted benzolactams are reported that are potent nonpeptidal antagonists of the peptide hormone cholecystokinin (CCK). Design considerations were based upon the natural product CCK antagonist asperlicin and the potent benzodiazepine a