10433-88-2Relevant articles and documents
NUCLEOPHILIC RING OPENING OF DIETHYL 1,1-CYCLOPROPANEDICARBOXYLATE USING Na2Fe(CO)4*3/2 DIOXANE
Tamblyn, William H.,Waltermire, Robert E.
, p. 2803 - 2806 (1983)
Diethyl 1,1-cyclopropanedicarboxylate undergoes nucleophilic ring opening with Na2Fe(CO)4*3/2 dioxane under CO at room temperature to produce a variety of carbonylated products.
BENZOQUINOLONE INHIBITORS OF VMAT2
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Paragraph 00117; 00118, (2015/04/15)
The present invention relates to new benzoquinolone inhibitors of VMAT2, pharmaceutical compositions thereof, and methods of use thereof represented by structural Formula I.
BENZOQUINOLINE INHIBITORS OF VESICULAR MONOAMINE TRANSPORTER 2
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Paragraph 00184; 00185, (2015/06/08)
The present invention relates to new benzoquinoline inhibitors of vesicular monoamine transporter 2 (VMAT2), pharmaceutical compositions thereof, and methods of use thereof. (I)
Phosphine-boronates: Efficient bifunctional organocatalysts for Michael addition
Basle, Olivier,Porcel, Susana,Ladeira, Sonia,Bouhadir, Ghenwa,Bourissou, Didier
supporting information; experimental part, p. 4495 - 4497 (2012/05/31)
Phosphine-boronates R2P(o-C6H4) B(OR′)2 have been evaluated as bifunctional organocatalysts for the Michael addition of malonate pronucleophiles to methylvinylketone. The presence of the Lewis acidic boron center adjacent to phosphorus significantly improves catalytic performance. Isolation and complete characterization of a key intermediate, namely a β-phosphonium enolate, substantiate the role of the Lewis acidic moiety in the catalytic process.