1428555-18-3Relevant articles and documents
Deconstruction of sulfonamide inhibitors of the urotensin receptor (UT) and design and synthesis of benzylamine and benzylsulfone antagonists
Taylor, Steven J.,Soleymanzadeh, Fariba,Muegge, Ingo,Akiba, Isamu,Taki, Naoyuki,Ueda, Saisoku,Mainolfi, Elizabeth,Eldrup, Anne B.
, p. 2177 - 2180 (2013/04/24)
Potent small molecule antagonists of the urotensin receptor are described. These inhibitors were derived via systematically deconstructing a literature inhibitor to understand the basic pharmacophore and key molecular features required to inhibit the prot
