259222-20-3Relevant articles and documents
Towards small molecule inhibitors of mono-ADP-ribosyltransferases
Ekblad, Torun,Lindgren, Anders E.G.,Andersson, C. David,Caraballo, Rémi,Thorsell, Ann-Gerd,Karlberg, Tobias,Spjut, Sara,Linusson, Anna,Schüler, Herwig,Elofsson, Mikael
supporting information, p. 546 - 551 (2015/04/14)
Protein ADP-ribosylation is a post-translational modification involved in DNA repair, protein degradation, transcription regulation, and epigenetic events. Intracellular ADP-ribosylation is catalyzed predominantly by ADP-ribosyltransferases with diphtheri