475630-67-2Relevant articles and documents
LACK OF GLYCOSIDASE INHIBITION BY, AND ISOLATION FROM XANTHOCERCIS ZAMBESIACA (LEGUMINOSAE) OF, 4-O-(&β-D-GLUCOPYRANOSYL)-FAGOMINE , A NOVEL GLUCOSIDE OF POLYHYDROXYLATED PIPERIDINE ALKALOID
Evans, Stephen V.,Hayman, Alison R.,Fellows, Linda E.,Shing, Tony K. M.,Derome, Andrew E.,Fleet, George W. J.
, p. 1465 - 1468 (1985)
A COSY spectrum has been used to determine the position of inter-residue linkage in 4-O-(β-D-glucopyranosyl) fagomine (1) an example of a new class of glycosides of polyhydroxylated piperidine alkaloids isolated from seed of the legume Xanthocercis zambesiaca. (Bak.) Dunn.Unlike a number of polyhydroxylated piperidines, neither the glucoside (1) nor the fagomine (3) showed any inhibitory activity towards glycosidase enzymes from a variety of sources.
N-Containing sugars from Morus alba and their glycosidase inhibitory activities
Asano, Naoki,Oseki, Kengo,Tomioka, Emiko,Kizu, Haruhisa,Matsui, Katsuhiko
, p. 243 - 256 (1994)
The reexamination of N-containing sugars from the roots of Morus alba by improved purification procedures led to the isolation of eighteen N-containing sugars, including seven that were isolated from the leaves of Morus bombycis.These N-containing sugars
Organocatalyzed synthesis of (-)-4-epi-fagomine and the corresponding pipecolic acids
Marjanovic, Jasna,Ferjancic, Zorana,Saicic, Radomir N.
, p. 6784 - 6789 (2015/08/24)
The enantioselective synthesis of 4-epi-fagomine was accomplished starting from dioxanone and Cbz-protected benyzlamine, in 4 steps, with 18% overall yield. The key feature of this synthetic approach is the tactical combination of reactions: organocatalyz
A PROCESS FOR SYNTHESIS OF PIPERIDINE ALKALOIDS
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Paragraph 0046; 0047, (2015/11/27)
The present invention discloses a process for synthesis of piperidine alkaloids selected from fagomine, 4-epi-fagomine and nojirimycin from tri-O-benzyl-D-glucal or tri-O-benzyl-D-galactal.