51659-21-3Relevant articles and documents
Direct Imination of Chalcones with Aminimide; Formation of Aziridines
Ikeda, Isao,Machii, Yoshimitsu,Okahara, Mitsuo
, p. 650 - 651 (1980)
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Synthesis of aziridines by electrochemical oxidative annulation of chalcones with primary amines
Gu, Lijun,He, Yonghui,Li, Ganpeng,Zeng, Dongwen,Zhang, Lizhu
, (2021/12/01)
Synthesis of aziridines by electrochemical oxidative annulation of chalcone 1,3-diphenyl-2-propen-1-one with primary amines has been developed under external oxidant - and base-free conditions. The reaction constitutes a new transformation of chalcones with primary amines to aziridines, providing a complementary, simple, and environmentally friendly approach to the currently available methods. A reaction mechanism for this transformation has been proposed based on the cyclic voltammetry.
Aminopyridinium iodide as a NH transferring agent for the synthesis of 2-aroyl-3-aryl aziridines
Samimi, Heshmat A.,Momeni, Ahmad R.
, p. 2221 - 2225 (2015/10/19)
A new approach for the synthesis of N-H ketoaziridines is described. 1-aminopyridinium iodide as a NH transferring agent provides a straightforward access to the 2-aroyl-3-arylaziridines from the corresponding 1,3-diarylprop-2-en-1-one. A possible general mechanism involving the N-N ylide is proposed.