909036-44-8Relevant articles and documents
Potent 4-amino-5-azaindole factor VIIa inhibitors
Hu, Huiyong,Kolesnikov, Aleksandr,Riggs, Jennifer R.,Wesson, Kieron E.,Stephens, Robin,Leahy, Ellen M.,Shrader, William D.,Sprengeler, Paul A.,Green, Michael J.,Sanford, Ellen,Nguyen, Margaret,Gjerstad, Erik,Cabuslay, Ronnel,Young, Wendy B.
, p. 4567 - 4570 (2007/10/03)
The 4-amino-5-azaindole as an amidino-benzimidazole replacement is described. A series of potent and selective analogs were discovered and showed desirable ex vivo efficacy as measured by PT.