Varenicline tartrate

Varenicline tartrate

Varenicline tartrate

Min.Order / FOB Price:Get Latest Price

1 Kilogram

Negotiable

  • Min.Order :1 Kilogram
  • Purity: 99%
  • Payment Terms : L/C,T/T,,MoneyGram,Other

Keywords

Varenicline tartrate price Varenicline tartrate CAS 375815-87-5 Varenicline tartrate supplier in China

Quick Details

  • Appearance:tan solid
  • Application:Nicotinic a4? acetylcholine receptor partial agonist. Aid in smoking cessation.
  • PackAge:100g/bottle,1kg/bottle,25kg/drum or as per your request
  • ProductionCapacity:1|Metric Ton|Month
  • Storage:Stored in cool, dry and ventilation place; Away from fire and heat
  • Transportation:by sea or by air

Superiority:

 

supplier in China

Details:

 

 
Varenicline tartrate Usage And Synthesis
Chemical Properties Tan Solid
Usage Nicotinic a4? acetylcholine receptor partial agonist. Aid in smoking cessation.
Usage Nicotinic α4β2 acetylcholine receptor partial agonist. Aid in smoking cessation.
Usage Varenicline is a prescription medication used to treat smoking addiction. Varenicline is a nicotinic receptor partial agonist. In this respect, it is similar to cytisine and different from the nicotinic antagonist, bupropion, and nicotine replacement ther
Biological Activity Orally active, subtype-selective partial agonist at α 4 β 2 nicotinic receptors (K i values are 0.06, 240, 322 and 3540 nM for α 4 β 2, α 3 β 4, α 7, α 1 β γ δ receptors respectively). Reduces nicotine-evoked dopamine release in vitro and decreases nicotine self-administration in vivo .

 

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