WZ 811 N1,N4-Di-2-pyridinyl-1,4-benzenedimethanamine;WZ 811;N,N'-Di-2-pyridinyl-1,4-benzenedimethanamine;N,N'-(1,4-phenylenebis(methylene))bis(pyridin-2-amine);1,4-Benzenedimethanamine, N1,N4-di-2-pyridinyl- 55778-02-4
WZ811 is a novel small molecular and potency CXCR4 antagonist with EC50 of 0.3 nM.
IC50 Value: 0.3 nM(EC50)
Target: CXCR4
in vitro: WZ811 efficiently inhibits CXCR4/stromal cell-derived factor-1 (SDF-1)-mediated modulation of cyclic adenosine monophophate (cAMP) levels (EC50 = 1.2 nM) and SDF-1 induced Matrigel invasion (EC50 = 5.2 nM).
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