Testolone（RAD140） manufacturer 1182367-47-0 in stock low price 1182367-47-0

Testolone（RAD140） manufacturer 1182367-47-0 in stock low price 1182367-47-0

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Testolone（RAD140） manufacturer 1182367-47-0 in stock low price 1182367-47-0

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Appearance:White solid
Application:pharmaceutical intermediates
PackAge:1kg/Aluminum foil package, 25Kg/Drum
ProductionCapacity:|Metric Ton|Day
Storage:Normal temperature
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Testolone（RAD140） manufacturer 1182367-47-0 in stock low price 1182367-47-0

Testolone, also known as RAD140, is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and breast cancer, currently under development by Radius Health, Inc. (RDUS). RAD140 Inhibits the Growth of Androgen/Estrogen Receptor Positive Breast Cancer Models with a Distinct Mechanism of Action.

RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that demonstrates excellent affinity for the androgen receptor (Ki = 7 nM). It displays potent anabolic effects in rodents and non-human primates and good bioavailability. It also demonstrates neuroprotective properties in hippocampal neurons of rat kainite model.

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RAD140 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a K_i value of 7 nM. At 0.03-0.3 mg/kg, it has been shown to stimulate muscle weight increase without affecting prostate or seminal vesicle in castrated male rats. At 0.3-1 mg/kg, RAD140 demonstrates partial antagonist activity in seminal vesicle and prostate.

Catalogue Number	R020050
Chemical Name	RAD 140
Synonyms	2-Chloro-4-[[(1R,2S)-1-[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]-2-hydroxypropyl]amino]-3-methylbenzonitrile
CAS Number	1182367-47-0
Molecular Formula	C??H??ClN?O?
Appearance	White Solid
Melting Point	179-183ºC
Molecular Weight	393.83
Storage	-20°C Freezer
Solubility	Chloroform (Slightly), DMSO (Slightly)
Category	Standards; Enzyme Activators and Inhibitors; Neurochemicals;
Applications	RAD 140 is a potent, orally bio-available, and non-steroidal selective androgen receptor modulator (SARM).

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