tianeptine sulfate CAS 30123-17-2 Tianeptine sodium salt

Superiority:

Tianeptine sodium is a salt of Tianeptine. Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake . Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation.
 

Function:
Tianeptine sodium is antidepressant. The animal has: the hippocampus pyramidal cells increased spontaneous activity, and accelerating its function was inhibited after recovery; increase in cortical and hippocampal neurons at sites of 5- serotonin reuptake. Tianeptine without following adverse effects: sleep and alertness; cardiovascular system; cholinergic system ( without anticholinergic symptoms ); drug craving.

Product Name:Tianeptine sodium
Trade Name:Stablon,Coaxil
CAS No.: 30123-17-2
Molecular Formula: C21H24ClN2NaO4S
Molecular Weight: 458.93g/mol
Specifition: USP
Purity : 99% HPLC
Elimination half-life:2.5-3h
Appearance:  White to off-white powder
Application :Antidepressants
Standard Packing :10g,100g,1kg
Shelf Life :2 years
Storage:Room temperature away from light

Description:

Tianeptine sodium salt is a salt of Tianeptine. Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake and is similar to amineptie. Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation counter.
Raw Tianeptine sodium salt powder is an atypical antidepressant with diverse actions, most notably on the glutamatergic system.It attenuates glutamate release and modulates the function of the AMPA receptor.Tianeptine also acts as an agonist of the μ-opioid receptor (EC50s = 194 and 641 nM for human and mouse receptors, respectively). It is as effective as fluoxetine in the management of post-traumatic stress disorder.
Tianeptine sodium salt has nootropic abilities in regards to individuals whose cognition is negatively impacted by mood disorders and has the ability to improve focus and concentration in individuals who have poor attention spans as well.

 
Typical Properties: 

• Tianeptine sodium salt can treat major depressive disorder.
• Tianeptine sodium salt has anti-anxiety and antidepressant and  and nootropic qualities.
• Tianeptine sodium salt enhance mood and improve mental status.
• Tianeptine sodium salt could block panic attacks from occurring.
• Tianeptine sodium salt treat pain associated with fibromyalgia.
• Tianeptine sodium salt used in treatment of depression in men with dysfunction.
• Tianeptine sodium salt has mild efficacy for ADHD.
• Tianeptine sodium salt also promotes neuroplasticity.

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