Calmodulin antagoni...

Calmodulin antagonist-1

Calmodulin antagonist-1

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Negotiable

  • Min.Order :0
  • Purity: ≥95%

Keywords

N-(4-Aminobutyl)-5-chloro-1-naphthalenesulfonamide Hydrochloride W8 Hydrochloride

Quick Details

  • Appearance:Pale Yellow to Yellow Solid
  • Application:Neoplasm inhibitor.
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  • Storage:Store at -20°C
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Details:

Calmodulin antagonist-1 is a calmodulin (CaM) antagonist that inhibits calmodulin-activated Ca2+-phosphodiesterase (PDE) (IC50 = 28 μM). Calmodulin antagonist-1 also inhibits trypsin-treated Ca2+-PDE (IC50 = 375 μM) in a competitive fashion with respect to cyclic GMP (Ki = 300 μM).

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