LY-309887 N-((5-(2-((6R)-2-Amino-3,4,5,6,7,8-hexahydro-4-oxopyrido(2,3-d)pyrimidin-6-yl)ethyl)-2-thienyl)carbonyl)-L-glutamic acid
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LY309887 is a potent inhibitor of glycinamide ribonucleotide formyltransferase (GARFT) with a Ki of 6.5 nM, and has antitumor activity.
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