Plm IV inhibitor-1 N1-((2S,3R)-3-hydroxy-1-phenyl-4-((2-(pyridin-2-yl)propan-2-yl)amino)butan-2-yl)-5-(piperidin-1-yl)-N3,N3-dipropylisophthalamide
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PG394 is a potent plasmepsin IV (Plm IV) inhibitor with IC50s of 4.1, 0.80, 0.25, 0.35 μM for Plm I, Plm II, Plm IV, Cat D, respectively.
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