Add time:09/02/2019         Source:sciencedirect.com

Studies of the binding of [3H]-SKF10047 to rat brain membrane preparations revealed a binding site which possessed high affinity for κ and agonist/antagonist analgesics. However, this site was distinguished from κ sites labelled with [3H]-ethylketazocine by its high affinity for Met5-enkephalin Arg6. Phe7 and β-endorphin as well as its low affinity for dynorphin 1–13. We therefore tentatively suggest that this may represent a possible κ isoreceptor population.

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