1242185-14-3Relevant articles and documents
Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors
Bova, Floriana,Ettari, Roberta,Micale, Nicola,Carnovale, Caterina,Schirmeister, Tanja,Gelhaus, Christoph,Leippe, Matthias,Grasso, Silvana,Zappal, Maria
experimental part, p. 4928 - 4938 (2010/09/05)
Herein we report the synthesis of a series of novel constrained peptidomimetics 2-10 endowed with a dipeptide backbone (d-Ser-Gly) and a vinyl ester warhead, structurally related to a previously identified lead compound 1, an irreversible inhibitor of fal