1356544-07-4Relevant articles and documents
Synthesis and in vitro evaluation of 2-[11C]methoxyestradiol-3, 17β-O,O-bissulfamate for in vivo studies of angiogenesis
Kang, Choong Mo,Choe, Yearn Seong,Jung, Kyung-Ho,Choi, Joon Young,Lee, Kyung-Han,Kim, Byung-Tae
, p. 783 - 787 (2011)
In the present study, 2-methoxyestradiol-3,17β-O,O-bissulfamate (1), a known angiogenesis inhibitor, was prepared in a radiolabeled form by 11C-methylation of 2-hydroxyestradiol-3,17β-O,O-bis(N-trityl) sulfamate (6) followed by detritylation. S