118939-18-7Relevant articles and documents
Process Development and Scale-Up of a Benzoxazepine-Containing Kinase Inhibitor
Naganathan, Sriram,Andersen, Denise L.,Andersen, Neil G.,Lau, Stephen,Lohse, Anders,Sorensen, Mads Detlef
, p. 721 - 734 (2015/07/27)
The benzoxazepine core is present in several kinase inhibitors, including the mTOR inhibitor 1. The process development for a scalable synthesis of 7-bromobenzoxazepine and the telescoped synthesis of 1 are reported. Compound 1 consists of three chemicall
3-cyclopropyl-4-(3-amino-2-methylbenzoyl)pyrazoles and their use as herbicides
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Page/Page column 8, (2008/06/13)
What is described are 3-cyclopropyl-4-(3-amino-2-methylbenzoyl)pyrazoles of the formula (I) and their use as herbicides. In this formula (I), R1, R2, R3, R4 and R5 are various radicals.